Tetrahedron

Direct assembly of N-sulfamoyl lactam scaffolds bearing a zinc-binding group for inhibiting metalloenzymes based on desymmetrization of sulfamide and the Castagnoli-Cushman reaction

Pub Date : 2024-02-01 DOI: 10.1016/j.tet.2024.133890 Elizaveta Karchuganova, Sofiia Martynova, Stanislav Kalinin, A. Angeli, Dmitry Dar'in, Daniella Vullo, C. Supuran, O. Bakulina

Aminopyridinium ylides from pyrano[3,4-c]pyran-7-ium salts: Synthesis and structure

Pub Date : 2024-02-01 DOI: 10.1016/j.tet.2024.133891 Alexander А. Chekunov, Konstantin F. Suzdalev, Valery V. Tkachev, Alina V. Krachkovskaya, Leonid D. Popov, Sergey M. Aldoshin, P. Galenko-Yaroshevsky, Yuri V. Tovkach